| DB05478 | Pradefovir mesylate | investigational | unknown | | Details |
| DB00180 | Flunisolide | approved, investigational | unknown | substrateinducer | Details |
| DB00185 | Cevimeline | approved | unknown | substrate | Details |
| DB00188 | Bortezomib | approved, investigational | no | substrate | Details |
| DB00196 | Fluconazole | approved, investigational | unknown | inhibitor | Details |
| DB00204 | Dofetilide | approved, investigational | unknown | substrate | Details |
| DB00213 | Pantoprazole | approved | unknown | substrate | Details |
| DB00216 | Eletriptan | approved, investigational | unknown | substrate | Details |
| DB00220 | Nelfinavir | approved | no | substrateinhibitor | Details |
| DB00224 | Indinavir | approved | unknown | substrateinhibitor | Details |
| DB00227 | Lovastatin | approved, investigational | unknown | substrateinhibitor | Details |
| DB00234 | Reboxetine | approved, experimental | unknown | substrateinhibitor | Details |
| DB00238 | Nevirapine | approved | unknown | substrateinducer | Details |
| DB00243 | Ranolazine | approved, investigational | no | substrateinhibitor | Details |
| DB00246 | Ziprasidone | approved | unknown | substrate | Details |
| DB00270 | Isradipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00280 | Disopyramide | approved | unknown | substrate | Details |
| DB00286 | Conjugated estrogens | approved | no | substrate | Details |
| DB00294 | Etonogestrel | approved, investigational | no | substrate | Details |
| DB00297 | Bupivacaine | approved, investigational | unknown | substrate | Details |
| DB00307 | Bexarotene | approved, investigational | unknown | substrateinducer | Details |
| DB00309 | Vindesine | approved, investigational | unknown | substrate | Details |
| DB00317 | Gefitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00324 | Fluorometholone | approved, investigational | unknown | substrateinducer | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00343 | Diltiazem | approved, investigational | unknown | substrateinhibitor | Details |
| DB00346 | Alfuzosin | approved, investigational | unknown | substrate | Details |
| DB00361 | Vinorelbine | approved, investigational | no | substrate | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00370 | Mirtazapine | approved | unknown | substrateinhibitor | Details |
| DB00381 | Amlodipine | approved | no | substrate | Details |
| DB00393 | Nimodipine | approved, investigational | unknown | substrate | Details |
| DB00398 | Sorafenib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00401 | Nisoldipine | approved | unknown | substrate | Details |
| DB00402 | Eszopiclone | approved, investigational | unknown | substrate | Details |
| DB00404 | Alprazolam | approved, illicit, investigational | unknown | substrate | Details |
| DB00425 | Zolpidem | approved | unknown | substrate | Details |
| DB00443 | Betamethasone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00455 | Loratadine | approved, investigational | no | substrateinhibitor | Details |
| DB00468 | Quinine | approved | unknown | substrateinhibitorinducer | Details |
| DB00470 | Dronabinol | approved, illicit | no | substrateinhibitor | Details |
| DB00471 | Montelukast | approved | unknown | substrate | Details |
| DB00490 | Buspirone | approved, investigational | unknown | substrate | Details |
| DB00496 | Darifenacin | approved, investigational | unknown | substrate | Details |
| DB00518 | Albendazole | approved, vet_approved | unknown | substrate | Details |
| DB00528 | Lercanidipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00533 | Rofecoxib | approved, investigational, withdrawn | unknown | substrateinducer | Details |
| DB00539 | Toremifene | approved, investigational | unknown | substrateinhibitor | Details |
| DB00541 | Vincristine | approved, investigational | unknown | substrate | Details |
| DB00559 | Bosentan | approved, investigational | unknown | substrateinducer | Details |
| DB00570 | Vinblastine | approved | unknown | substrateinhibitorinducer | Details |
| DB00582 | Voriconazole | approved | unknown | substrateinhibitor | Details |
| DB00588 | Fluticasone propionate | approved | unknown | substrateinhibitor | Details |
| DB00593 | Ethosuximide | approved | unknown | substrate | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | unknown | substrateinducer | Details |
| DB00604 | Cisapride | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00615 | Rifabutin | approved, investigational | unknown | substrateinducer | Details |
| DB00619 | Imatinib | approved | no | substrateinhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrateinducer | Details |
| DB00625 | Efavirenz | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00635 | Prednisone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00636 | Clofibrate | approved, investigational | unknown | substrateinducer | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00641 | Simvastatin | approved | unknown | substrate | Details |
| DB00673 | Aprepitant | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00674 | Galantamine | approved | no | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrateinhibitorinducer | Details |
| DB00678 | Losartan | approved | unknown | substrateinhibitor | Details |
| DB00683 | Midazolam | approved, illicit | unknown | substrateinhibitor | Details |
| DB00696 | Ergotamine | approved | unknown | substrateinhibitor | Details |
| DB00700 | Eplerenone | approved | unknown | substrate | Details |
| DB00701 | Amprenavir | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00705 | Delavirdine | approved | unknown | substrateinhibitor | Details |
| DB00731 | Nateglinide | approved, investigational | unknown | substrate | Details |
| DB00736 | Esomeprazole | approved, investigational | unknown | substrate | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00744 | Zileuton | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00745 | Modafinil | approved, investigational | unknown | substrateinducer | Details |
| DB00757 | Dolasetron | approved, investigational | unknown | substrate | Details |
| DB00758 | Clopidogrel | approved | no | substrate | Details |
| DB00762 | Irinotecan | approved, investigational | unknown | substrateinhibitor | Details |
| DB00769 | Hydrocortamate | approved | unknown | inducer | Details |
| DB00773 | Etoposide | approved | unknown | substrateinhibitorinducer | Details |
| DB00778 | Roxithromycin | approved, investigational, withdrawn | no | substrateinhibitor | Details |
| DB00802 | Alfentanil | approved, illicit | unknown | substrate | Details |
| DB00813 | Fentanyl | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00820 | Tadalafil | approved, investigational | no | substrate | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00834 | Mifepristone | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00836 | Loperamide | approved | unknown | substrateinhibitor | Details |
| DB00843 | Donepezil | approved | unknown | substrate | Details |
| DB00860 | Prednisolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00862 | Vardenafil | approved | unknown | substrateinhibitor | Details |
| DB00864 | Tacrolimus | approved, investigational | unknown | substrate | Details |
| DB00872 | Conivaptan | approved, investigational | unknown | substrateinhibitor | Details |
| DB00877 | Sirolimus | approved, investigational | no | substrate | Details |
| DB00889 | Granisetron | approved, investigational | unknown | substrate | Details |
| DB00897 | Triazolam | approved, investigational | unknown | substrate | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | substrate | Details |
| DB00906 | Tiagabine | approved, investigational | unknown | substrate | Details |
| DB00907 | Cocaine | approved, illicit | unknown | substrate | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | substrate | Details |
| DB00910 | Paricalcitol | approved, investigational | unknown | substrate | Details |
| DB00911 | Tinidazole | approved, investigational | unknown | substrate | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00932 | Tipranavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB00938 | Salmeterol | approved | unknown | substrate | Details |
| DB00956 | Hydrocodone | approved, illicit, investigational | unknown | substrate | Details |
| DB00959 | Methylprednisolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00962 | Zaleplon | approved, illicit, investigational | unknown | substrate | Details |
| DB00976 | Telithromycin | approved | unknown | substrateinhibitor | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB00990 | Exemestane | approved, investigational | unknown | substrate | Details |
| DB00997 | Doxorubicin | approved, investigational | no | substrateinhibitor | Details |
| DB01002 | Levobupivacaine | approved, investigational | unknown | substrate | Details |
| DB01006 | Letrozole | approved, investigational | unknown | substrate | Details |
| DB01008 | Busulfan | approved, investigational | unknown | substrate | Details |
| DB01012 | Cinacalcet | approved | unknown | substrate | Details |
| DB01023 | Felodipine | approved, investigational | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB01054 | Nitrendipine | approved, investigational | unknown | substrate | Details |
| DB01062 | Oxybutynin | approved, investigational | unknown | substrateinhibitor | Details |
| DB01068 | Clonazepam | approved, illicit | unknown | substrate | Details |
| DB01072 | Atazanavir | approved, investigational | no | substrateinhibitor | Details |
| DB01076 | Atorvastatin | approved | no | substrate | Details |
| DB01100 | Pimozide | approved | unknown | substrate | Details |
| DB01105 | Sibutramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB01114 | Chlorpheniramine | approved | unknown | substrate | Details |
| DB01115 | Nifedipine | approved | unknown | substrateinhibitorinducer | Details |
| DB01129 | Rabeprazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB01132 | Pioglitazone | approved, investigational | unknown | substrateinducer | Details |
| DB01149 | Nefazodone | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB01166 | Cilostazol | approved, investigational | unknown | substrate | Details |
| DB01167 | Itraconazole | approved, investigational | no | substrateinhibitor | Details |
| DB01175 | Escitalopram | approved | no | substrate | Details |
| DB01184 | Domperidone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01190 | Clindamycin | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | no | substrateinhibitor | Details |
| DB01206 | Lomustine | approved, investigational | unknown | inhibitor | Details |
| DB01211 | Clarithromycin | approved | unknown | substrateinhibitor | Details |
| DB01215 | Estazolam | approved, illicit | unknown | substrate | Details |
| DB01216 | Finasteride | approved | unknown | substrate | Details |
| DB01218 | Halofantrine | approved | unknown | substrate | Details |
| DB01222 | Budesonide | approved | no | substrateinducer | Details |
| DB01224 | Quetiapine | approved | unknown | substrate | Details |
| DB01227 | Levacetylmethadol | approved, investigational, withdrawn | unknown | substrate | Details |
| DB01229 | Paclitaxel | approved, vet_approved | unknown | substrateinducer | Details |
| DB01232 | Saquinavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB01238 | Aripiprazole | approved, investigational | no | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01256 | Retapamulin | approved | unknown | substrate | Details |
| DB01261 | Sitagliptin | approved, investigational | unknown | substrate | Details |
| DB01259 | Lapatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01264 | Darunavir | approved | unknown | substrateinhibitor | Details |
| DB01268 | Sunitinib | approved, investigational | no | substrateinhibitor | Details |
| DB01263 | Posaconazole | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | inducer | Details |
| DB01601 | Lopinavir | approved | unknown | substrateinhibitor | Details |
| DB01411 | Pranlukast | investigational | no | substrate | Details |
| DB01410 | Ciclesonide | approved, investigational | no | substrate | Details |
| DB00969 | Alosetron | approved, withdrawn | unknown | substrate | Details |
| DB04835 | Maraviroc | approved, investigational | unknown | substrate | Details |
| DB01409 | Tiotropium | approved | unknown | substrate | Details |
| DB01591 | Solifenacin | approved | no | substrate | Details |
| DB01011 | Metyrapone | approved, investigational | unknown | inhibitorinducer | Details |
| DB00377 | Palonosetron | approved, investigational | unknown | substrate | Details |
| DB04856 | Dexloxiglumide | investigational | unknown | substrate | Details |
| DB04886 | Calanolide A | investigational | unknown | substrate | Details |
| DB00580 | Valdecoxib | approved, investigational, withdrawn | unknown | substrate | Details |
| DB06144 | Sertindole | approved, investigational, withdrawn | unknown | substrate | Details |
| DB04977 | Plitidepsin | investigational | unknown | substrate | Details |
| DB04905 | Tesmilifene | investigational | unknown | substrateinhibitorinducer | Details |
| DB00333 | Methadone | approved | unknown | substrateinhibitorinducer | Details |
| DB04934 | Rifalazil | investigational | unknown | substrate | Details |
| DB04957 | Azimilide | investigational | unknown | substrate | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | no | substrateinhibitor | Details |
| DB01628 | Etoricoxib | approved, investigational | unknown | substrateinhibitor | Details |
| DB00564 | Carbamazepine | approved, investigational | unknown | substrateinducer | Details |
| DB06155 | Rimonabant | approved, investigational | unknown | substrate | Details |
| DB06267 | Udenafil | approved, investigational | unknown | substrate | Details |
| DB06287 | Temsirolimus | approved | unknown | substrate | Details |
| DB06442 | Avasimibe | investigational | unknown | inducer | Details |
| DB08502 | Capravirine | investigational | unknown | substrate | Details |
| DB06652 | Vicriviroc | investigational | unknown | substrate | Details |
| DB06685 | Laquinimod | investigational | unknown | substrate | Details |
| DB01095 | Fluvastatin | approved | unknown | substrateinhibitor | Details |
| DB00203 | Sildenafil | approved, investigational | unknown | substrate | Details |
| DB00248 | Cabergoline | approved | unknown | substrate | Details |
| DB00589 | Lisuride | approved, investigational | unknown | substrate | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB05271 | Rotigotine | approved | unknown | substrate | Details |
| DB00439 | Cerivastatin | approved, withdrawn | unknown | substrateinhibitorinducer | Details |
| DB00257 | Clotrimazole | approved, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB00734 | Risperidone | approved, investigational | unknown | substrate | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB01037 | Selegiline | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | substrate | Details |
| DB01181 | Ifosfamide | approved | unknown | substrateinhibitorinducer | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00814 | Meloxicam | approved, vet_approved | unknown | substrate | Details |
| DB00908 | Quinidine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00656 | Trazodone | approved, investigational | unknown | substrate | Details |
| DB00176 | Fluvoxamine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB00540 | Nortriptyline | approved | unknown | substrate | Details |
| DB00215 | Citalopram | approved | no | substrateinhibitor | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | substrate | Details |
| DB00472 | Fluoxetine | approved, vet_approved | no | substrateinhibitor | Details |
| DB01104 | Sertraline | approved | unknown | substrateinhibitor | Details |
| DB06148 | Mianserin | approved, investigational | unknown | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB01118 | Amiodarone | approved, investigational | no | substrateinhibitor | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrateinducer | Details |
| DB05109 | Trabectedin | approved, investigational | unknown | substrate | Details |
| DB00946 | Phenprocoumon | approved, investigational | unknown | substrate | Details |
| DB00682 | Warfarin | approved | unknown | substrateinducer | Details |
| DB00285 | Venlafaxine | approved | unknown | substrate | Details |
| DB00857 | Terbinafine | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB00972 | Azelastine | approved | unknown | substrateinhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | substrateinhibitor | Details |
| DB00661 | Verapamil | approved | unknown | substrateinhibitor | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | substrateinducer | Details |
| DB00201 | Caffeine | approved | unknown | substrate | Details |
| DB00318 | Codeine | approved, illicit | unknown | substrate | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | substrateinhibitor | Details |
| DB00502 | Haloperidol | approved | unknown | substrateinhibitor | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | substrate | Details |
| DB00571 | Propranolol | approved, investigational | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00446 | Chloramphenicol | approved, vet_approved, withdrawn | unknown | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | unknown | inhibitor | Details |
| DB01059 | Norfloxacin | approved | unknown | inhibitor | Details |
| DB06403 | Ambrisentan | approved, investigational | unknown | substrate | Details |
| DB06413 | Armodafinil | approved, investigational | unknown | inducer | Details |
| DB00865 | Benzphetamine | approved, illicit | unknown | substrate | Details |
| DB00612 | Bisoprolol | approved | unknown | substrate | Details |
| DB00136 | Calcitriol | approved, nutraceutical | unknown | substrateinducer | Details |
| DB00608 | Chloroquine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | no | substrateinducer | Details |
| DB00628 | Clorazepic acid | approved, illicit | unknown | substrate | Details |
| DB01396 | Digitoxin | approved, investigational | unknown | substrate | Details |
| DB04855 | Dronedarone | approved | unknown | substrateinhibitor | Details |
| DB04574 | Estrone sulfate | approved | unknown | substrate | Details |
| DB06414 | Etravirine | approved | unknown | substrateinducer | Details |
| DB01590 | Everolimus | approved | unknown | substrate | Details |
| DB00949 | Felbamate | approved | unknown | substrateinducer | Details |
| DB06702 | Fesoterodine | approved | unknown | substrate | Details |
| DB00690 | Flurazepam | approved, illicit, investigational | unknown | substrate | Details |
| DB00499 | Flutamide | approved, investigational | unknown | substrate | Details |
| DB01018 | Guanfacine | approved, investigational | unknown | substrate | Details |
| DB04845 | Ixabepilone | approved, investigational | unknown | substrate | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB00367 | Levonorgestrel | approved, investigational | unknown | substrate | Details |
| DB00358 | Mefloquine | approved, investigational | unknown | substrateinhibitor | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB00497 | Oxycodone | approved, illicit, investigational | unknown | substrate | Details |
| DB06589 | Pazopanib | approved | unknown | substrateinhibitor | Details |
| DB01621 | Pipotiazine | approved, investigational | unknown | substrate | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | no | substrate | Details |
| DB01087 | Primaquine | approved | unknown | substrateinhibitor | Details |
| DB00647 | Dextropropoxyphene | approved, illicit, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00912 | Repaglinide | approved, investigational | unknown | substrate | Details |
| DB06228 | Rivaroxaban | approved | unknown | substrate | Details |
| DB06176 | Romidepsin | approved, investigational | unknown | substrate | Details |
| DB06207 | Silodosin | approved | unknown | substrate | Details |
| DB00706 | Tamsulosin | approved, investigational | unknown | substrate | Details |
| DB00444 | Teniposide | approved | unknown | substrateinhibitor | Details |
| DB00759 | Tetracycline | approved, vet_approved, withdrawn | unknown | substrateinhibitor | Details |
| DB00277 | Theophylline | approved | unknown | substrate | Details |
| DB01036 | Tolterodine | approved, investigational | unknown | substrate | Details |
| DB06212 | Tolvaptan | approved | unknown | substrate | Details |
| DB00193 | Tramadol | approved, investigational | unknown | substrate | Details |
| DB00440 | Trimethoprim | approved, vet_approved | unknown | substrate | Details |
| DB01198 | Zopiclone | approved | unknown | substrate | Details |
| DB00357 | Aminoglutethimide | approved, investigational | unknown | inducer | Details |
| DB01320 | Fosphenytoin | approved, investigational | unknown | substrateinducer | Details |
| DB00607 | Nafcillin | approved, investigational | unknown | inducer | Details |
| DB00776 | Oxcarbazepine | approved | unknown | inhibitorinducer | Details |
| DB00312 | Pentobarbital | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrateinducer | Details |
| DB00794 | Primidone | approved, vet_approved | unknown | inducer | Details |
| DB01201 | Rifapentine | approved, investigational | unknown | substrateinducer | Details |
| DB01394 | Colchicine | approved | unknown | substrateinhibitor | Details |
| DB01253 | Ergometrine | approved | unknown | substrate | Details |
| DB01221 | Ketamine | approved, vet_approved | unknown | substrateinducer | Details |
| DB00353 | Methylergometrine | approved | unknown | substrateinhibitor | Details |
| DB06335 | Saxagliptin | approved | unknown | substrate | Details |
| DB00708 | Sufentanil | approved, investigational | unknown | substrate | Details |
| DB01128 | Bicalutamide | approved | unknown | substrateinhibitor | Details |
| DB01151 | Desipramine | approved, investigational | unknown | inhibitor | Details |
| DB00916 | Metronidazole | approved | unknown | inhibitor | Details |
| DB06268 | Sitaxentan | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrateinhibitorinducer | Details |
| DB00420 | Promazine | approved, vet_approved | unknown | substrate | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | substrateinhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB00482 | Celecoxib | approved, investigational | unknown | substrate | Details |
| DB01016 | Glyburide | approved | unknown | substrateinhibitor | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | substrateinducer | Details |
| DB06739 | Seratrodast | experimental | unknown | substrateinducer | Details |
| DB06738 | Ketobemidone | investigational | unknown | substrate | Details |
| DB01242 | Clomipramine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00655 | Estrone | approved | no | substrate | Details |
| DB00458 | Imipramine | approved | unknown | substrate | Details |
| DB00546 | Adinazolam | experimental | unknown | substrate | Details |
| DB00231 | Temazepam | approved, investigational | unknown | substrate | Details |
| DB03701 | Vanoxerine | investigational | unknown | substrate | Details |
| DB00169 | Cholecalciferol | approved, nutraceutical | unknown | substrate | Details |
| DB01192 | Oxymorphone | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01173 | Orphenadrine | approved | unknown | substrateinhibitor | Details |
| DB06772 | Cabazitaxel | approved | unknown | substrate | Details |
| DB02709 | Resveratrol | investigational | no | inhibitor | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | substrateinhibitor | Details |
| DB06697 | Artemether | approved | unknown | substrateinducer | Details |
| DB06708 | Lumefantrine | approved | unknown | substrate | Details |
| DB00819 | Acetazolamide | approved, vet_approved | unknown | inhibitor | Details |
| DB06742 | Ambroxol | approved, investigational | unknown | substrate | Details |
| DB01223 | Aminophylline | approved | unknown | substrate | Details |
| DB00278 | Argatroban | approved, investigational | unknown | substrate | Details |
| DB01169 | Arsenic trioxide | approved, investigational | unknown | inhibitor | Details |
| DB00207 | Azithromycin | approved | unknown | substrateinhibitor | Details |
| DB01393 | Bezafibrate | approved, investigational | unknown | substrate | Details |
| DB04794 | Bifonazole | approved, investigational | unknown | inhibitor | Details |
| DB01194 | Brinzolamide | approved | no | substrate | Details |
| DB00520 | Caspofungin | approved | unknown | inhibitor | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00356 | Chlorzoxazone | approved | unknown | substrateinhibitor | Details |
| DB00845 | Clofazimine | approved, investigational | unknown | inhibitor | Details |
| DB06470 | Clomethiazole | investigational | unknown | substrate | Details |
| DB01559 | Clotiazepam | approved, illicit | unknown | substrate | Details |
| DB00987 | Cytarabine | approved, investigational | unknown | substrate | Details |
| DB01406 | Danazol | approved | unknown | inhibitor | Details |
| DB00694 | Daunorubicin | approved | unknown | substrateinhibitor | Details |
| DB01093 | Dimethyl sulfoxide | approved, vet_approved | unknown | inhibitor | Details |
| DB00822 | Disulfiram | approved | unknown | substrate | Details |
| DB00254 | Doxycycline | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB01127 | Econazole | approved | no | inhibitor | Details |
| DB00751 | Epinastine | approved, investigational | unknown | substrate | Details |
| DB00668 | Epinephrine | approved, vet_approved | unknown | inhibitor | Details |
| DB01196 | Estramustine | approved, investigational | unknown | substrate | Details |
| DB00898 | Ethanol | approved | unknown | substrateinhibitorinducer | Details |
| DB01466 | Ethylmorphine | experimental, illicit | unknown | substrate | Details |
| DB00301 | Flucloxacillin | approved, investigational | unknown | substrateinducer | Details |
| DB01544 | Flunitrazepam | approved, illicit | unknown | substrate | Details |
| DB00947 | Fulvestrant | approved, investigational | unknown | substrate | Details |
| DB01275 | Hydralazine | approved | no | inhibitor | Details |
| DB00724 | Imiquimod | approved, investigational | unknown | substrate | Details |
| DB01029 | Irbesartan | approved, investigational | no | inhibitor | Details |
| DB00602 | Ivermectin | approved, investigational, vet_approved | no | substrate | Details |
| DB01103 | Quinacrine | investigational | unknown | substrate | Details |
| DB01071 | Mequitazine | experimental | unknown | inhibitor | Details |
| DB04817 | Metamizole | approved, investigational, withdrawn | unknown | inducer | Details |
| DB04833 | Methaqualone | illicit, withdrawn | unknown | substrate | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | unknown | substrate | Details |
| DB06710 | Methyltestosterone | approved | unknown | substrate | Details |
| DB00379 | Mexiletine | approved, investigational | unknown | substrate | Details |
| DB01204 | Mitoxantrone | approved, investigational | unknown | inhibitor | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | substrateinhibitor | Details |
| DB02701 | Nicotinamide | approved, investigational | unknown | inhibitor | Details |
| DB00184 | Nicotine | approved | unknown | substrate | Details |
| DB01595 | Nitrazepam | approved | unknown | substrate | Details |
| DB00768 | Olopatadine | approved | no | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrateinducer | Details |
| DB01074 | Perhexiline | approved, investigational | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrate | Details |
| DB00454 | Meperidine | approved | unknown | substrateinducer | Details |
| DB03783 | Phenacetin | withdrawn | unknown | substrate | Details |
| DB00780 | Phenelzine | approved | unknown | inhibitor | Details |
| DB00812 | Phenylbutazone | approved, vet_approved | unknown | inducer | Details |
| DB01085 | Pilocarpine | approved, investigational | unknown | inhibitor | Details |
| DB01588 | Prazepam | approved, illicit | unknown | substrate | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inducer | Details |
| DB01182 | Propafenone | approved | unknown | substrate | Details |
| DB01589 | Quazepam | approved, illicit | no | substrate | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | inhibitor | Details |
| DB00863 | Ranitidine | approved, withdrawn | unknown | inhibitor | Details |
| DB01220 | Rifaximin | approved, investigational | unknown | substrateinducer | Details |
| DB00296 | Ropivacaine | approved | unknown | substrate | Details |
| DB01698 | Rutin | approved, experimental, investigational | unknown | inducer | Details |
| DB01001 | Salbutamol | approved, vet_approved | unknown | inhibitor | Details |
| DB01236 | Sevoflurane | approved, vet_approved | unknown | substrate | Details |
| DB00359 | Sulfadiazine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01015 | Sulfamethoxazole | approved | unknown | substrate | Details |
| DB01349 | Tasosartan | experimental | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | inhibitor | Details |
| DB04572 | Thiotepa | approved, investigational | unknown | substrate | Details |
| DB01007 | Tioconazole | approved | unknown | inhibitor | Details |
| DB00273 | Topiramate | approved | unknown | inducer | Details |
| DB00347 | Trimethadione | approved | unknown | substrate | Details |
| DB13179 | Troleandomycin | approved | unknown | substrateinhibitor | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | inhibitor | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00495 | Zidovudine | approved | unknown | substrate | Details |
| DB04828 | Zomepirac | withdrawn | unknown | substrate | Details |
| DB01380 | Cortisone acetate | approved, investigational | unknown | substrateinducer | Details |
| DB01384 | Paramethasone | experimental | unknown | substrateinhibitorinducer | Details |
| DB01587 | Ketazolam | approved | unknown | substrateinhibitor | Details |
| DB08811 | Tofisopam | experimental | unknown | inhibitor | Details |
| DB00617 | Paramethadione | approved | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB00980 | Ramelteon | approved, investigational | unknown | substrate | Details |
| DB04946 | Iloperidone | approved | unknown | substrate | Details |
| DB01418 | Acenocoumarol | approved, investigational | unknown | substrate | Details |
| DB06684 | Vilazodone | approved | unknown | substrate | Details |
| DB00255 | Diethylstilbestrol | approved, investigational, withdrawn | unknown | substrateinhibitor | Details |
| DB00575 | Clonidine | approved | unknown | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | inhibitor | Details |
| DB00400 | Griseofulvin | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00808 | Indapamide | approved | unknown | substrate | Details |
| DB05521 | Telaprevir | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB08820 | Ivacaftor | approved | no | substrateinhibitor | Details |
| DB06634 | Casopitant | investigational | unknown | | Details |
| DB04975 | Banoxantrone | investigational | unknown | substrate | Details |
| DB05039 | Indacaterol | approved | unknown | substrate | Details |
| DB08816 | Ticagrelor | approved | unknown | substrateinhibitor | Details |
| DB06774 | Capsaicin | approved | unknown | inhibitor | Details |
| DB06174 | Noscapine | approved, investigational | unknown | inhibitor | Details |
| DB01333 | Cefradine | approved | unknown | inducer | Details |
| DB06777 | Chenodeoxycholic acid | approved | unknown | substrate | Details |
| DB00856 | Chlorphenesin | approved, experimental | unknown | inducer | Details |
| DB04920 | Clevidipine | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB01764 | Dalfopristin | approved | unknown | inhibitor | Details |
| DB01609 | Deferasirox | approved, investigational | unknown | inducer | Details |
| DB00485 | Dicloxacillin | approved, investigational, vet_approved | unknown | inducer | Details |
| DB06370 | Indisulam | investigational | unknown | inhibitor | Details |
| DB01083 | Orlistat | approved, investigational | unknown | inducer | Details |
| DB00239 | Oxiconazole | approved | unknown | inducer | Details |
| DB00082 | Pegvisomant | approved | unknown | inducer | Details |
| DB06762 | Pinacidil | approved | unknown | substrate | Details |
| DB01369 | Quinupristin | approved | unknown | inhibitor | Details |
| DB00337 | Pimecrolimus | approved, investigational | unknown | substrate | Details |
| DB00041 | Aldesleukin | approved | unknown | inhibitor | Details |
| DB06605 | Apixaban | approved | no | substrate | Details |
| DB08827 | Lomitapide | approved, investigational | no | substrate | Details |
| DB08828 | Vismodegib | approved, investigational | no | substrate | Details |
| DB00620 | Triamcinolone | approved, vet_approved | unknown | substrateinducer | Details |
| DB08864 | Rilpivirine | approved | no | substrateinhibitorinducer | Details |
| DB06209 | Prasugrel | approved | no | substrate | Details |
| DB06216 | Asenapine | approved | unknown | substrate | Details |
| DB00435 | Nitric Oxide | approved | unknown | inhibitor | Details |
| DB08867 | Ulipristal | approved | no | substrate | Details |
| DB08815 | Lurasidone | approved, investigational | unknown | substrate | Details |
| DB08870 | Brentuximab vedotin | approved, investigational | no | substrateinhibitor | Details |
| DB04871 | Lorcaserin | approved, withdrawn | no | substrate | Details |
| DB05294 | Vandetanib | approved | unknown | substrate | Details |
| DB08873 | Boceprevir | approved, withdrawn | unknown | substrateinhibitor | Details |
| DB08875 | Cabozantinib | approved, investigational | no | substrate | Details |
| DB08877 | Ruxolitinib | approved | unknown | substrate | Details |
| DB05812 | Abiraterone | approved | unknown | substrateinhibitor | Details |
| DB08881 | Vemurafenib | approved | unknown | substrateinducer | Details |
| DB08882 | Linagliptin | approved | unknown | substrateinhibitor | Details |
| DB08883 | Perampanel | approved | no | substrateinducer | Details |
| DB08865 | Crizotinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB06626 | Axitinib | approved, investigational | no | substrate | Details |
| DB08893 | Mirabegron | approved | no | substrate | Details |
| DB06237 | Avanafil | approved | unknown | substrate | Details |
| DB08896 | Regorafenib | approved | unknown | substrateinhibitor | Details |
| DB08899 | Enzalutamide | approved | no | substrateinducer | Details |
| DB08895 | Tofacitinib | approved, investigational | no | substrate | Details |
| DB06616 | Bosutinib | approved | no | substrateinhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | substrate | Details |
| DB08903 | Bedaquiline | approved | no | substrate | Details |
| DB06201 | Rufinamide | approved | unknown | inducer | Details |
| DB08906 | Fluticasone furoate | approved | no | substrateinhibitorinducer | Details |
| DB08907 | Canagliflozin | approved | unknown | substrate | Details |
| DB06203 | Alogliptin | approved | unknown | substrate | Details |
| DB04938 | Ospemifene | approved, investigational | unknown | substrate | Details |
| DB08910 | Pomalidomide | approved | unknown | substrate | Details |
| DB08911 | Trametinib | approved | unknown | substrateinducer | Details |
| DB08912 | Dabrafenib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB05773 | Trastuzumab emtansine | approved, investigational | unknown | substrate | Details |
| DB08833 | Taurochenodeoxycholic acid | experimental | unknown | substrate | Details |
| DB01142 | Doxepin | approved, investigational | no | substrate | Details |
| DB00688 | Mycophenolate mofetil | approved, investigational | unknown | substrate | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB08932 | Macitentan | approved | no | substrate | Details |
| DB08933 | Luliconazole | approved | no | inhibitor | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB09039 | Eliglustat | approved, investigational | no | substrate | Details |
| DB05676 | Apremilast | approved, investigational | no | substrate | Details |
| DB09049 | Naloxegol | approved | unknown | substrate | Details |
| DB09053 | Ibrutinib | approved | unknown | substrate | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | | Details |
| DB09074 | Olaparib | approved | unknown | substrateinhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB09073 | Palbociclib | approved, investigational | no | substrateinhibitor | Details |
| DB09054 | Idelalisib | approved | no | substrateinhibitorinducer | Details |
| DB09068 | Vortioxetine | approved, investigational | no | substrate | Details |
| DB09082 | Vilanterol | approved | no | substrate | Details |
| DB09083 | Ivabradine | approved | no | substrate | Details |
| DB09026 | Aliskiren | approved, investigational | no | substrate | Details |
| DB09101 | Elvitegravir | approved | no | substrateinhibitor | Details |
| DB06016 | Cariprazine | approved, investigational | no | substrateinhibitorinducer | Details |
| DB08439 | Parecoxib | approved | unknown | substrate | Details |
| DB09128 | Brexpiprazole | approved, investigational | no | substrate | Details |
| DB09291 | Rolapitant | approved, investigational | no | substrate | Details |
| DB04908 | Flibanserin | approved, investigational | no | substrate | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | substrate | Details |
| DB09143 | Sonidegib | approved, investigational | unknown | substrate | Details |
| DB06636 | Isavuconazonium | approved, investigational | no | substrateinhibitorinducer | Details |
| DB06603 | Panobinostat | approved, investigational | unknown | substrate | Details |
| DB05239 | Cobimetinib | approved, investigational | no | substrateinhibitor | Details |
| DB09570 | Ixazomib | approved, investigational | unknown | substrate | Details |
| DB09330 | Osimertinib | approved | no | substrateinhibitorinducer | Details |
| DB11362 | Selexipag | approved | no | substrate | Details |
| DB09119 | Eslicarbazepine acetate | approved | no | inducer | Details |
| DB06789 | Hydroxyprogesterone caproate | approved, investigational | unknown | substrate | Details |
| DB08931 | Riociguat | approved | unknown | substrate | Details |
| DB09183 | Dasabuvir | approved | no | substrate | Details |
| DB09297 | Paritaprevir | approved, investigational | no | substrate | Details |
| DB09317 | Synthetic Conjugated Estrogens, A | approved | no | substrate | Details |
| DB09318 | Synthetic Conjugated Estrogens, B | approved | no | substrate | Details |
| DB09389 | Norgestrel | approved | unknown | substrate | Details |
| DB11581 | Venetoclax | approved, investigational | no | substrateinhibitor | Details |
| DB09280 | Lumacaftor | approved | no | inducer | Details |
| DB01323 | St. John's Wort | approved, investigational, nutraceutical | unknown | substrateinduceractivator | Details |
| DB09381 | Esterified estrogens | approved | unknown | substrate | Details |
| DB00957 | Norgestimate | approved, investigational | unknown | substrateinducer | Details |
| DB04911 | Oritavancin | approved, investigational | unknown | inhibitorinducer | Details |
| DB06717 | Fosaprepitant | approved | unknown | substrateinhibitorinducer | Details |
| DB00648 | Mitotane | approved | unknown | inducer | Details |
| DB08909 | Glycerol phenylbutyrate | approved | unknown | inducer | Details |
| DB09048 | Netupitant | approved, investigational | no | substrateinhibitor | Details |
| DB12332 | Rucaparib | approved, investigational | no | substrateinhibitor | Details |
| DB11921 | Deflazacort | approved, investigational | no | substrateinducer | Details |
| DB11737 | Icotinib | experimental, investigational | unknown | substrate | Details |
| DB06654 | Safinamide | approved, investigational | unknown | substrate | Details |
| DB12161 | Deutetrabenazine | approved, investigational | no | substrate | Details |
| DB09555 | Dexchlorpheniramine maleate | approved | unknown | substrate | Details |
| DB11613 | Velpatasvir | approved, investigational | no | substrate | Details |
| DB05541 | Brivaracetam | approved, investigational | no | substrate | Details |
| DB11915 | Valbenazine | approved, investigational | no | substrate | Details |
| DB06670 | Odanacatib | investigational | no | substrate | Details |
| DB05351 | Dexlansoprazole | approved, investigational | unknown | substrate | Details |
| DB06290 | Simeprevir | approved | unknown | substrateinhibitor | Details |
| DB11575 | Grazoprevir | approved | no | substrateinhibitor | Details |
| DB11943 | Delafloxacin | approved, investigational | unknown | inducer | Details |
| DB01685 | Topiroxostat | experimental | unknown | inhibitor | Details |
| DB08922 | Perospirone | experimental | unknown | substrate | Details |
| DB09118 | Stiripentol | approved | unknown | substrateinhibitorinducer | Details |
| DB09166 | Etizolam | experimental | unknown | substrate | Details |
| DB11614 | Rupatadine | approved | no | substrate | Details |
| DB09262 | Imidafenacin | investigational | no | substrate | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | | Details |
| DB09238 | Manidipine | approved, investigational | unknown | substrateinhibitor | Details |
| DB09123 | Dienogest | approved | unknown | substrate | Details |
| DB11828 | Neratinib | approved, investigational | unknown | substrate | Details |
| DB12026 | Voxilaprevir | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | inhibitor | Details |
| DB00503 | Ritonavir | approved, investigational | unknown | substrateinhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB11574 | Elbasvir | approved | unknown | substrate | Details |
| DB12483 | Copanlisib | approved, investigational | no | substrate | Details |
| DB11767 | Sarilumab | approved, investigational | no | inhibitorinducer | Details |
| DB12001 | Abemaciclib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | no | substrate | Details |
| DB11817 | Baricitinib | approved, investigational | unknown | substrate | Details |
| DB13074 | Macimorelin | approved, investigational | unknown | substrate | Details |
| DB09223 | Blonanserin | investigational | no | substrate | Details |
| DB09236 | Lacidipine | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | substrateinhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrateinhibitorinducer | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrateinhibitorinducer | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB13952 | Estradiol acetate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB13953 | Estradiol benzoate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB13954 | Estradiol cypionate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB13955 | Estradiol dienanthate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB13956 | Estradiol valerate | approved, investigational, vet_approved | unknown | substrateinducer | Details |
| DB13941 | Piperaquine | approved, experimental, investigational | unknown | substrateinhibitor | Details |
| DB01420 | Testosterone propionate | approved, investigational, vet_approved, withdrawn | no | substrate | Details |
| DB09195 | Lorpiprazole | approved | no | substrate | Details |
| DB11799 | Bictegravir | approved, investigational | unknown | substrate | Details |
| DB11901 | Apalutamide | approved, investigational | no | substrateinducer | Details |
| DB09225 | Zotepine | approved, investigational, withdrawn | no | substrate | Details |
| DB09230 | Azelnidipine | investigational | unknown | substrate | Details |
| DB09231 | Benidipine | experimental | no | substrateinhibitor | Details |
| DB09235 | Efonidipine | experimental | unknown | substrateinhibitor | Details |
| DB11642 | Pitolisant | approved, investigational | unknown | substrateinducer | Details |
| DB11633 | Isavuconazole | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB09237 | Levamlodipine | approved, investigational | unknown | substrate | Details |
| DB11712 | Tezacaftor | approved, investigational | no | substrateinhibitorinducer | Details |
| DB11130 | Opium | approved, illicit | no | substrate | Details |
| DB11251 | Tocopherol | approved, investigational | no | substrate | Details |
| DB14003 | alpha-Tocopherol acetate | approved | no | substrate | Details |
| DB11586 | Asunaprevir | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB13975 | Black cohosh | experimental | no | inhibitor | Details |
| DB12278 | Propiverine | approved, investigational | no | substrate | Details |
| DB14011 | Nabiximols | investigational | unknown | substrate | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |
| DB11641 | Vinflunine | approved, investigational | no | substrate | Details |
| DB11635 | Tocofersolan | approved | no | substrate | Details |
| DB11637 | Delamanid | approved, investigational | no | substrate | Details |
| DB13746 | Bioallethrin | approved, experimental | no | substrate | Details |
| DB14019 | Fosnetupitant | approved | unknown | substrateinhibitor | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01049 | Ergoloid mesylate | approved | no | substrate | Details |
| DB11274 | Dihydro-alpha-ergocryptine | approved | no | substrate | Details |
| DB13293 | Ipecac | approved, withdrawn | no | substrate | Details |
| DB11198 | Peppermint oil | approved, investigational | unknown | inhibitor | Details |
| DB13456 | Midecamycin | experimental | no | substrateinhibitor | Details |
| DB12532 | Oxetacaine | approved, investigational | no | inhibitor | Details |
| DB11672 | Curcumin | approved, investigational | unknown | inhibitor | Details |
| DB11779 | Danoprevir | investigational | no | inhibitor | Details |
| DB09289 | Tianeptine | investigational | no | substrate | Details |
| DB01357 | Mestranol | approved | no | substrate | Details |
| DB04829 | Lysergic acid diethylamide | illicit, investigational, withdrawn | no | substrate | Details |
| DB00247 | Methysergide | approved | no | substrate | Details |
| DB13399 | Terguride | experimental | no | substrate | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | substrate | Details |
| DB11718 | Encorafenib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB14538 | Hydrocortisone aceponate | experimental, vet_approved | unknown | substrateinducer | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14541 | Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | substrate | Details |
| DB14542 | Hydrocortisone phosphate | approved, vet_approved | unknown | substrate | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14568 | Ivosidenib | approved, investigational | unknown | substrateinducer | Details |
| DB12629 | 3,5-diiodothyropropionic acid | investigational | no | substrate | Details |
| DB01456 | 5-androstenedione | experimental, illicit | no | substrate | Details |
| DB00240 | Alclometasone | approved | no | substrate | Details |
| DB04630 | Aldosterone | experimental, investigational | no | substrate | Details |
| DB00288 | Amcinonide | approved | no | substrateinducer | Details |
| DB01536 | Androstenedione | experimental, illicit | no | substrate | Details |
| DB00394 | Beclomethasone dipropionate | approved, investigational | no | substrateinducer | Details |
| DB11750 | Clobetasol | approved, experimental, investigational | no | substrateinducer | Details |
| DB01013 | Clobetasol propionate | approved | no | substrateinducer | Details |
| DB13158 | Clobetasone | approved | no | substrate | Details |
| DB04652 | Corticosterone | experimental | no | substrate | Details |
| DB01285 | Corticotropin | approved, investigational, vet_approved | no | substrateinducer | Details |
| DB04839 | Cyproterone acetate | approved, investigational | no | substrateinhibitor | Details |
| DB11636 | Nomegestrol | approved | no | substrate | Details |
| DB13981 | Nomegestrol acetate | approved, investigational | no | substrate | Details |
| DB00304 | Desogestrel | approved | no | substrate | Details |
| DB01260 | Desonide | approved, investigational | no | substrateinducer | Details |
| DB06780 | Desoxycorticosterone acetate | approved | no | substrate | Details |
| DB01134 | Desoxycorticosterone pivalate | experimental, vet_approved | no | substrate | Details |
| DB11487 | Dexamethasone isonicotinate | vet_approved | no | substrateinhibitorinducer | Details |
| DB09095 | Difluocortolone | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB06781 | Difluprednate | approved | no | substrate | Details |
| DB00378 | Dydrogesterone | approved, investigational, withdrawn | no | substrate | Details |
| DB03515 | Equilenin | experimental | no | substrate | Details |
| DB02187 | Equilin | experimental | no | substrate | Details |
| DB13866 | Etynodiol | experimental | no | substrate | Details |
| DB00823 | Ethynodiol diacetate | approved | no | substrate | Details |
| DB00687 | Fludrocortisone | approved, investigational | unknown | substrate | Details |
| DB00663 | Flumethasone | approved, vet_approved | no | substrate | Details |
| DB00591 | Fluocinolone acetonide | approved, investigational, vet_approved | no | substrateinducer | Details |
| DB01047 | Fluocinonide | approved, investigational | no | substrateinducer | Details |
| DB08971 | Fluocortolone | approved, withdrawn | no | substrateinducer | Details |
| DB08970 | Fluprednidene | experimental | no | substrateinducer | Details |
| DB09378 | Fluprednisolone | approved | no | substrate | Details |
| DB00846 | Flurandrenolide | approved | no | substrate | Details |
| DB13867 | Fluticasone | approved, experimental | no | substrateinhibitorinducer | Details |
| DB08905 | Formestane | approved, investigational, withdrawn | no | inducer | Details |
| DB06730 | Gestodene | investigational | no | substrateinhibitor | Details |
| DB11619 | Gestrinone | approved | no | substrate | Details |
| DB06786 | Halcinonide | approved, investigational, withdrawn | no | substrate | Details |
| DB05212 | HE3286 | investigational | no | substrate | Details |
| DB14545 | Hydrocortisone succinate | approved | unknown | substrateinducer | Details |
| DB14570 | Hydroxyprogesterone | experimental | no | substrate | Details |
| DB01583 | Liotrix | approved | no | substrate | Details |
| DB14596 | Loteprednol etabonate | approved | unknown | substrate | Details |
| DB12474 | Lynestrenol | approved, investigational | no | substrate | Details |
| DB09124 | Medrogestone | approved, withdrawn | no | substrate | Details |
| DB00253 | Medrysone | approved | no | substrateinducer | Details |
| DB00351 | Megestrol acetate | approved, investigational, vet_approved | no | substrate | Details |
| DB11529 | Melengestrol | vet_approved | no | substrate | Details |
| DB09383 | Meprednisone | approved, investigational | no | substrateinducer | Details |
| DB00764 | Mometasone | experimental | no | substrateinducer | Details |
| DB14512 | Mometasone furoate | approved, investigational, vet_approved | no | substrateinducer | Details |
| DB06713 | Norelgestromin | approved, investigational | no | substrate | Details |
| DB09371 | Norethynodrel | approved | no | substrate | Details |
| DB01130 | Prednicarbate | approved, investigational | no | substrate | Details |
| DB13208 | Prednylidene | experimental | no | substrateinducer | Details |
| DB02789 | Pregnenolone | approved, experimental | no | substrate | Details |
| DB13602 | Promegestone | experimental | no | substrate | Details |
| DB00896 | Rimexolone | approved | no | substrateinducer | Details |
| DB01117 | Atovaquone | approved | no | substrate | Details |
| DB11753 | Rifamycin | approved, investigational | no | inhibitorinducer | Details |
| DB13528 | Chlormadinone | experimental | no | substrate | Details |
| DB13857 | Demegestone | experimental | no | substrate | Details |
| DB13685 | Quingestanol | experimental | no | substrate | Details |
| DB14055 | (S)-Warfarin | experimental, investigational | no | substrate | Details |
| DB13347 | Diphenadione | experimental | no | substrate | Details |
| DB08794 | Ethyl biscoumacetate | withdrawn | unknown | substrate | Details |
| DB01483 | Barbital | illicit | no | inducer | Details |
| DB01154 | Thiamylal | approved, vet_approved | no | substrateinducer | Details |
| DB09229 | Aranidipine | experimental | no | substrate | Details |
| DB09227 | Barnidipine | experimental | no | substrateinhibitor | Details |
| DB13488 | Bencyclane | experimental | no | substrate | Details |
| DB01244 | Bepridil | approved, withdrawn | no | substrate | Details |
| DB08838 | Agmatine | experimental | no | substrate | Details |
| DB11960 | Carboxyamidotriazole | investigational | no | substrate | Details |
| DB13835 | Caroverine | experimental | no | substrate | Details |
| DB09232 | Cilnidipine | investigational | no | substrate | Details |
| DB00568 | Cinnarizine | approved, investigational | no | substrate | Details |
| DB04838 | Cyclandelate | approved | no | substrate | Details |
| DB09234 | Darodipine | experimental | no | substrate | Details |
| DB14068 | Dexniguldipine | experimental | no | substrate | Details |
| DB14063 | Dexverapamil | experimental | no | substrate | Details |
| DB06446 | Dotarizine | investigational | no | substrate | Details |
| DB14064 | Emopamil | experimental | no | substrate | Details |
| DB08992 | Eperisone | investigational | no | substrate | Details |
| DB08980 | Fendiline | withdrawn | no | substrate | Details |
| DB13961 | Fish oil | approved, nutraceutical | no | substrate | Details |
| DB04841 | Flunarizine | approved | no | substrate | Details |
| DB04842 | Fluspirilene | approved, investigational | no | substrate | Details |
| DB12923 | Gallopamil | investigational | no | substrate | Details |
| DB13766 | Lidoflazine | approved, experimental | no | substrate | Details |
| DB14065 | Lomerizine | experimental | no | substrate | Details |
| DB00825 | Levomenthol | approved | no | substrate | Details |
| DB12092 | Naftopidil | investigational | no | substrate | Details |
| DB09239 | Niguldipine | experimental | no | substrate | Details |
| DB09240 | Niludipine | experimental | no | substrate | Details |
| DB04743 | Nimesulide | approved, investigational, withdrawn | no | substrate | Details |
| DB06152 | Nylidrin | approved | no | substrate | Details |
| DB13500 | Otilonium | experimental, investigational | no | substrate | Details |
| DB13791 | Penfluridol | experimental | no | substrate | Details |
| DB09090 | Pinaverium | approved | no | substrate | Details |
| DB04825 | Prenylamine | approved, withdrawn | no | substrate | Details |
| DB13725 | Terodiline | experimental | no | substrate | Details |
| DB12093 | Tetrahydropalmatine | investigational | no | substrate | Details |
| DB14066 | Tetrandrine | experimental | no | substrate | Details |
| DB09216 | Tolfenamic acid | approved, investigational | no | substrate | Details |
| DB07615 | Tranilast | investigational | no | substrate | Details |
| DB09089 | Trimebutine | approved | no | substrate | Details |
| DB05885 | Seletracetam | investigational | no | substrate | Details |
| DB12131 | Vinpocetine | investigational | no | substrate | Details |
| DB13950 | WIN 55212-2 | experimental | no | substrateinhibitor | Details |
| DB04070 | 6-Deoxyerythronolide B | experimental | no | inhibitor | Details |
| DB06318 | AVE9633 | investigational | no | inhibitor | Details |
| DB07348 | Brefeldin A | experimental | no | inhibitor | Details |
| DB11752 | Bryostatin 1 | investigational | no | inhibitor | Details |
| DB01152 | Candicidin | approved, withdrawn | no | inhibitor | Details |
| DB11383 | Carbomycin | vet_approved | no | inhibitor | Details |
| DB06419 | Cethromycin | investigational | no | substrateinhibitor | Details |
| DB06342 | Coltuximab ravtansine | investigational | no | inhibitor | Details |
| DB00954 | Dirithromycin | experimental | no | inhibitor | Details |
| DB11400 | Doramectin | vet_approved | no | inhibitor | Details |
| DB12266 | Epofolate | investigational | no | inhibitor | Details |
| DB01873 | Epothilone D | investigational | no | inhibitor | Details |
| DB11405 | Eprinomectin | vet_approved | no | inhibitor | Details |
| DB13338 | Flurithromycin | experimental | no | inhibitor | Details |
| DB05814 | GPI-1485 | investigational | no | inhibitor | Details |
| DB09309 | Kitasamycin | experimental | no | inhibitor | Details |
| DB05903 | KOS-1584 | investigational | no | inhibitor | Details |
| DB12089 | Lorvotuzumab mertansine | investigational | no | inhibitor | Details |
| DB13287 | Miocamycin | approved | no | inhibitor | Details |
| DB12489 | Mirvetuximab soravtansine | approved, investigational | no | substrateinhibitor | Details |
| DB06587 | Mitemcinal | investigational | no | inhibitor | Details |
| DB11442 | Oleandomycin | vet_approved | no | inhibitor | Details |
| DB03010 | Patupilone | experimental, investigational | no | inhibitor | Details |
| DB06233 | Ridaforolimus | investigational | no | inhibitor | Details |
| DB13409 | Rokitamycin | experimental | no | inhibitor | Details |
| DB12391 | Sagopilone | investigational | no | inhibitor | Details |
| DB11459 | Selamectin | vet_approved | no | inhibitor | Details |
| DB09308 | Solithromycin | investigational | no | inhibitor | Details |
| DB11470 | Tildipirosin | vet_approved | no | inhibitor | Details |
| DB01241 | Gemfibrozil | approved | unknown | substrate | Details |
| DB06791 | Lanreotide | approved | no | inhibitor | Details |
| DB00104 | Octreotide | approved, investigational | no | inhibitor | Details |
| DB06663 | Pasireotide | approved | no | inhibitor | Details |
| DB09099 | Somatostatin | approved, investigational | no | inhibitor | Details |
| DB04894 | Vapreotide | experimental, investigational | no | inhibitor | Details |
| DB12781 | Balaglitazone | investigational | no | substrate | Details |
| DB09201 | Ciglitazone | experimental | no | substrate | Details |
| DB09198 | Lobeglitazone | experimental | no | substrate | Details |
| DB09199 | Netoglitazone | experimental | no | substrate | Details |
| DB09200 | Rivoglitazone | experimental, investigational | no | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | no | substrateinducer | Details |
| DB09063 | Ceritinib | approved | no | substrateinhibitor | Details |
| DB06469 | Lestaurtinib | investigational | no | inhibitor | Details |
| DB11805 | Saracatinib | investigational | no | inhibitor | Details |
| DB11703 | Acalabrutinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB01267 | Paliperidone | approved | unknown | substrate | Details |
| DB01645 | Genistein | investigational | unknown | inducer | Details |
| DB05928 | Dovitinib | investigational | unknown | inhibitor | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB11919 | 6-O-benzylguanine | investigational | no | substrate | Details |
| DB14583 | Segesterone acetate | approved, experimental, investigational | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | no | substrate | Details |
| DB04884 | Dapoxetine | investigational | no | substrateinhibitor | Details |
| DB08953 | Indalpine | investigational, withdrawn | no | substrateinhibitor | Details |
| DB00715 | Paroxetine | approved, investigational | no | substrateinhibitor | Details |
| DB04832 | Zimelidine | approved, withdrawn | no | inhibitor | Details |
| DB04896 | Milnacipran | approved, investigational | no | substrateinhibitor | Details |
| DB02703 | Fusidic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB11730 | Ribociclib | approved, investigational | no | substrateinhibitor | Details |
| DB09079 | Nintedanib | approved | no | substrate | Details |
| DB14634 | Fluprednidene acetate | experimental | no | inducer | Details |
| DB14637 | Fluprednisolone acetate | experimental | no | substrate | Details |
| DB01656 | Roflumilast | approved | no | substrate | Details |
| DB09034 | Suvorexant | approved, investigational | no | substrate | Details |
| DB09071 | Tasimelteon | approved, investigational | no | substrate | Details |
| DB09030 | Vorapaxar | approved | no | substrate | Details |
| DB01624 | Zuclopenthixol | approved, investigational | no | substrate | Details |
| DB13385 | Dihydroergocryptine | experimental | no | substrate | Details |
| DB11273 | Dihydroergocornine | approved | no | substrate | Details |
| DB13345 | Dihydroergocristine | approved, experimental | no | substrate | Details |
| DB06218 | Lacosamide | approved | no | substrate | Details |
| DB12329 | Eravacycline | approved, investigational | unknown | substrate | Details |
| DB06458 | Remacemide | investigational | no | inhibitor | Details |
| DB08874 | Fidaxomicin | approved | no | inhibitor | Details |
| DB11742 | Ebastine | approved, investigational | no | substrate | Details |
| DB09036 | Siltuximab | approved, investigational | no | inducer | Details |
| DB06273 | Tocilizumab | approved | no | inducer | Details |
| DB12301 | Doravirine | approved, investigational | unknown | substrate | Details |
| DB11952 | Duvelisib | approved, investigational | no | substrate | Details |
| DB13997 | Baloxavir marboxil | approved, investigational | no | substrateinhibitor | Details |
| DB00186 | Lorazepam | approved | no | substrate | Details |
| DB12515 | 9-aminocamptothecin | investigational | no | substrate | Details |
| DB12952 | Methylprednisone | approved, investigational | no | substrate | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | substrate | Details |
| DB11963 | Dacomitinib | approved, investigational | no | substrate | Details |
| DB12141 | Gilteritinib | approved, investigational | no | substrate | Details |
| DB14723 | Larotrectinib | approved, investigational | no | substrate | Details |
| DB12537 | 1,2-Benzodiazepine | approved, investigational | unknown | substrate | Details |
| DB09017 | Brotizolam | investigational, withdrawn | unknown | substrate | Details |
| DB11094 | Vitamin D | approved, nutraceutical, vet_approved | no | substrate | Details |
| DB01352 | Aprobarbital | experimental, illicit | unknown | inducer | Details |
| DB00590 | Doxazosin | approved | no | substrate | Details |
| DB05482 | SN-38 | investigational | unknown | substrateinhibitor | Details |
| DB06480 | Prucalopride | approved | no | substrate | Details |
| DB11978 | Glasdegib | approved, investigational | no | substrate | Details |
| DB12582 | Piperine | investigational | unknown | inhibitor | Details |
| DB00191 | Phentermine | approved, illicit | no | substrate | Details |
| DB12245 | Triclabendazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB00264 | Metoprolol | approved, investigational | no | substrate | Details |
| DB11823 | Esketamine | approved, investigational | unknown | substrateinducer | Details |
| DB00163 | Vitamin E | approved, nutraceutical, vet_approved | unknown | substrateinducer | Details |
| DB12371 | Siponimod | approved, investigational | unknown | substrate | Details |
| DB12147 | Erdafitinib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB09299 | Tenofovir alafenamide | approved | no | substrate | Details |
| DB00982 | Isotretinoin | approved | unknown | substrate | Details |
| DB12015 | Alpelisib | approved, investigational | unknown | substrate | Details |
| DB12240 | Polatuzumab vedotin | approved, investigational | no | substrate | Details |
| DB00905 | Bimatoprost | approved, investigational | unknown | substrate | Details |
| DB11942 | Selinexor | approved, investigational | unknown | substrate | Details |
| DB14669 | Betamethasone phosphate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14652 | Clocortolone acetate | experimental | unknown | inducer | Details |
| DB13843 | Cloprednol | experimental | unknown | inducer | Details |
| DB14681 | Cortisone | experimental | unknown | inducer | Details |
| DB13003 | Cortivazol | investigational | unknown | inducer | Details |
| DB13728 | Halometasone | experimental | unknown | inducer | Details |
| DB14659 | Melengestrol acetate | experimental | unknown | inducer | Details |
| DB14644 | Methylprednisolone hemisuccinate | approved | unknown | inducer | Details |
| DB14633 | Prednisolone hemisuccinate | experimental | unknown | inducer | Details |
| DB14631 | Prednisolone phosphate | approved, vet_approved | unknown | substrateinducer | Details |
| DB14646 | Prednisone acetate | approved, experimental, investigational | unknown | inducer | Details |
| DB02520 | Ditiocarb | experimental | unknown | inhibitor | Details |
| DB06731 | Seproxetine | investigational | unknown | inhibitor | Details |
| DB00627 | Niacin | approved, investigational, nutraceutical | unknown | inhibitor | Details |
| DB06282 | Levocetirizine | approved | unknown | substrate | Details |
| DB09173 | Butyrfentanyl | illicit | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB01551 | Dihydrocodeine | approved, illicit | unknown | substrate | Details |
| DB05154 | Pretomanid | approved | unknown | substrate | Details |
| DB01395 | Drospirenone | approved | unknown | substrate | Details |
| DB01611 | Hydroxychloroquine | approved | unknown | substrate | Details |
| DB11986 | Entrectinib | approved, investigational | unknown | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | substrate | Details |
| DB12825 | Lefamulin | approved, investigational | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB01319 | Fosamprenavir | approved | unknown | substrateinhibitor | Details |
| DB01050 | Ibuprofen | approved | no | substrate | Details |
| DB15489 | Mexazolam | experimental | unknown | substrate | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | inhibitor | Details |
| DB09288 | Propacetamol | experimental | unknown | substrateinducer | Details |
| DB01233 | Metoclopramide | approved, investigational | unknown | substrate | Details |
| DB11761 | Tenapanor | approved, investigational | unknown | substrate | Details |
| DB14635 | Curcumin sulfate | experimental | unknown | inhibitor | Details |
| DB14600 | Edetate disodium anhydrous | approved, vet_approved | unknown | inhibitor | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrateinhibitor | Details |
| DB14575 | Eslicarbazepine | approved | unknown | inducer | Details |
| DB12808 | Trifarotene | approved, investigational | unknown | substrate | Details |
| DB15444 | Elexacaftor | approved, investigational | no | substrateinhibitor | Details |
| DB15566 | Prednisolone acetate | approved, vet_approved | unknown | substrateinducer | Details |
| DB00557 | Hydroxyzine | approved | no | substrate | Details |
| DB14240 | Echinacea | approved, experimental | unknown | inducer | Details |
| DB11560 | Lesinurad | approved, investigational | unknown | inducer | Details |
| DB15035 | Zanubrutinib | approved, investigational | no | substrate | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | unknown | inhibitorinducer | Details |
| DB13879 | Glecaprevir | approved, investigational | unknown | inhibitor | Details |
| DB14975 | Voxelotor | approved, investigational | unknown | substrate | Details |
| DB00717 | Norethisterone | approved | unknown | substrate | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB13007 | Enfortumab vedotin | approved, investigational | unknown | substrate | Details |
| DB14962 | Trastuzumab deruxtecan | approved, investigational | unknown | substrate | Details |
| DB11951 | Lemborexant | approved, investigational | unknown | substrate | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | substrate | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB15091 | Upadacitinib | approved, investigational | no | substrate | Details |
| DB15328 | Ubrogepant | approved, investigational | unknown | substrate | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | substrate | Details |
| DB12887 | Tazemetostat | approved, investigational | unknown | substrate | Details |
| DB12457 | Rimegepant | approved, investigational | no | substrateinhibitor | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | substrateinhibitor | Details |
| DB14678 | Norethindrone enanthate | experimental | unknown | substrate | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB12612 | Ozanimod | approved, investigational | unknown | substrate | Details |
| DB14598 | Edetate calcium disodium anhydrous | approved | unknown | inhibitor | Details |
| DB11689 | Selumetinib | approved, investigational | no | substrate | Details |
| DB15102 | Pemigatinib | approved, investigational | no | substrate | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | substrateinhibitor | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | substrate | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | substrate | Details |
| DB14840 | Ripretinib | approved | unknown | substrate | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | | Details |
| DB12674 | Lurbinectedin | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | substrateinhibitorinducer | Details |
| DB00574 | Fenfluramine | approved, illicit, investigational, withdrawn | unknown | substrate | Details |
| DB05015 | Belinostat | approved, investigational | unknown | substrate | Details |
| DB11796 | Fostemsavir | approved, investigational | unknown | substrate | Details |
| DB11932 | Abametapir | approved, investigational | no | inhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB14881 | Oliceridine | approved, investigational | no | substrate | Details |
| DB12499 | Clascoterone | approved, investigational | no | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB06448 | Lonafarnib | approved, investigational | unknown | substrateinhibitor | Details |
| DB15982 | Berotralstat | approved | no | inhibitor | Details |
| DB06137 | Tirbanibulin | approved, investigational | no | substrateinhibitor | Details |
| DB14895 | Vibegron | approved, investigational | no | substrate | Details |
| DB00475 | Chlordiazepoxide | approved, illicit, investigational | unknown | substrate | Details |
| DB00752 | Tranylcypromine | approved, investigational | unknown | inhibitor | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | no | substrateinhibitorinducer | Details |
| DB00476 | Duloxetine | approved | unknown | inhibitor | Details |
| DB11693 | Voclosporin | approved, investigational | unknown | substrateinhibitor | Details |
| DB15133 | Tepotinib | approved, investigational | no | substrateinhibitor | Details |
| DB00747 | Scopolamine | approved, investigational | no | substrate | Details |
| DB00330 | Ethambutol | approved | unknown | inhibitor | Details |
| DB14989 | Umbralisib | approved, investigational, withdrawn | unknown | substrate | Details |
| DB14984 | Casimersen | approved, investigational | no | inhibitor | Details |
| DB00545 | Pyridostigmine | approved, investigational | no | inducer | Details |
| DB11800 | Tivozanib | approved, investigational | unknown | substrate | Details |
| DB12016 | Ponesimod | approved, investigational | unknown | substrate | Details |
| DB08995 | Diosmin | approved, investigational | unknown | inhibitor | Details |
| DB05316 | Pimavanserin | approved, investigational | unknown | substrate | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB12235 | Estetrol | approved, investigational | unknown | substrate | Details |
| DB16222 | Loncastuximab tesirine | approved, investigational | unknown | | Details |
| DB11886 | Infigratinib | approved, investigational | no | substrate | Details |
| DB12471 | Ibrexafungerp | approved, investigational | unknown | substrateinhibitor | Details |
| DB12543 | Samidorphan | approved, investigational | no | substrate | Details |
| DB16165 | Finerenone | approved, investigational | unknown | substrate | Details |
| DB16703 | Belumosudil | approved, investigational | no | substrate | Details |
| DB12130 | Lorlatinib | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB15463 | Belzutifan | approved, investigational | no | substrate | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrateinhibitor | Details |
| DB16390 | Mobocertinib | approved, investigational | unknown | substrate | Details |
| DB16732 | Tisotumab vedotin | approved | no | substrate | Details |
| DB16098 | Atogepant | approved, investigational | no | substrate | Details |
| DB16226 | Maralixibat | approved, investigational | no | inhibitor | Details |
| DB15011 | Avacopan | approved, investigational | no | substrateinhibitorinducer | Details |
| DB12597 | Asciminib | approved, investigational | no | substrateinhibitor | Details |
| DB06234 | Maribavir | approved, investigational | no | substrate | Details |
| DB16691 | Nirmatrelvir | approved, investigational | no | substrateinhibitor | Details |
| DB15031 | Daridorexant | approved | no | substrate | Details |
| DB12713 | Sotagliflozin | approved, investigational | no | substrateinhibitorinducer | Details |
| DB14973 | Abrocitinib | approved, investigational | no | substrate | Details |
| DB05467 | Palovarotene | approved, investigational | no | substrateinducer | Details |
| DB16236 | Mitapivat | approved, investigational | no | substrateinducer | Details |
| DB12834 | Secnidazole | approved | unknown | substrateinhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | unknown | substrateinhibitor | Details |
| DB00486 | Nabilone | approved, investigational | unknown | substrateinhibitor | Details |
| DB06230 | Nalmefene | approved, investigational, withdrawn | no | substrate | Details |
| DB11697 | Pacritinib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB05087 | Ganaxolone | approved, investigational | no | substrate | Details |
| DB01041 | Thalidomide | approved, investigational, withdrawn | no | substrateinducer | Details |
| DB14921 | Mavacamten | approved, investigational | no | substrateinducer | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | inhibitor | Details |
| DB00951 | Isoniazid | approved, investigational | unknown | inhibitor | Details |
| DB12020 | Tecovirimat | approved, investigational | no | inducer | Details |
| DB06083 | Tapinarof | approved, investigational | no | substrate | Details |
| DB01024 | Mycophenolic acid | approved, investigational | unknown | substrate | Details |
| DB10534 | Grapefruit | approved | unknown | inhibitor | Details |
| DB04951 | Pirfenidone | approved, investigational | unknown | inhibitor | Details |
| DB15673 | Lenacapavir | approved, investigational | no | substrateinhibitor | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inhibitorinducer | Details |
| DB15149 | Futibatinib | approved, investigational | no | substrate | Details |
| DB17083 | Linzagolix | approved | no | substrate | Details |
| DB11739 | Vonoprazan | approved, investigational | unknown | substrate | Details |
| DB09065 | Cobicistat | approved | yes | inhibitor | Details |
| DB16267 | Olutasidenib | approved, investigational | no | substrateinducer | Details |
| DB15568 | Adagrasib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12236 | Bexagliflozin | approved, investigational | unknown | substrate | Details |
| DB17472 | Pirtobrutinib | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB06374 | Elacestrant | approved, investigational | unknown | substrate | Details |
| DB11682 | Daprodustat | approved, investigational | no | substrate | Details |
| DB09065 | Cobicistat | approved | no | substrate | Details |
| DB12548 | Sparsentan | approved, investigational | unknown | substrateinhibitorinducer | Details |
| DB12513 | Omaveloxolone | approved, investigational | unknown | substrateinducer | Details |
| DB15688 | Zavegepant | approved, investigational | unknown | substrate | Details |
| DB06045 | Trofinetide | approved, investigational | unknown | inhibitor | Details |
| DB16217 | Leniolisib | approved, investigational | no | substrate | Details |
| DB12255 | Vadadustat | approved, investigational | unknown | downregulator | Details |
| DB14924 | Ritlecitinib | approved, investigational | unknown | substrateinhibitor | Details |
| DB12874 | Quizartinib | approved, investigational | no | substrate | Details |
| DB15490 | Zuranolone | approved, experimental | no | substrate | Details |
| DB11763 | Momelotinib | approved, investigational | unknown | substrate | Details |
| DB12184 | Gepirone | approved, investigational | no | substrate | Details |
| DB14766 | Etrasimod | approved | no | substrate | Details |
| DB15114 | Vamorolone | approved, investigational | no | substrateinducer | Details |
| DB12218 | Capivasertib | approved, investigational | no | substrate | Details |
| DB16826 | Repotrectinib | approved, investigational | no | substrateinhibitorinducer | Details |
| DB11679 | Fruquintinib | approved, investigational | no | substrate | Details |
| DB12005 | Nirogacestat | approved, investigational | no | substrate | Details |
| DB11995 | Avatrombopag | approved, investigational | no | substrate | Details |